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Anti-Androgens

Our Anti-Androgens class of Mens Health medications are used to block the action of testosterone in certain conditions including treating androgen-dependent prostate cancer and to treat hypersexuality.

Use the search feature to quickly find the product you are looking for, by entering either the active ingredient, e.g. cyproterone or the product name, e.g. Siterone.

What is an anti-androgen?

Anti-androgens are drugs that counteract the biological effects of the male hormone testosterone or its active metabolite DHT. They bind to the same androgen receptor as testosterone in specific cells and act as androgen receptor antagonists because they block the biological action of testosterone and DHT working through this receptor. Anti-androgens are either steroidal or non-steroidal and act in a competitive manner for the receptors.

Steroidal anti-androgens

Cyproterone is a steroidal anti-androgen that binds to the androgen receptor competing with testosterone and blocking testosterone binding to its receptor. However, cyproterone does have some biological effects, acting as a weak progestogen and glucocorticoid, which are other hormones involved in production of sex hormones like testosterone. This means that cyproterone does not prevent the production of testosterone completely but reduces the amount of testosterone produced. Cyproterone is used to treat hypersexuality (increased sex drive) and aggression in male sex offenders. It is also used to treat advanced prostate cancer.

Non-steroidal anti-androgens

Bicalutamide is a non-steroidal anti-androgen that binds to the androgen receptor but has no androgen or any other hormonal activity. It does not activate any normal testosterone actions, which means that it does not promote prostate cell growth or testosterone production. Bicalutamide is used to treat advanced prostate cancer, in combination with another medication that induces medical castration by preventing testosterone production by the testes. This blocks the stimulation by testosterone of cancer cell growth and helps slow or prevent progression of the tumour.
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Stevie Rhodes UK • May 2025
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Robert Lypka NC, USA • June 2025
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Dave MI, USA • May 2026
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"Hello, just a quick message to compliment you & your staff on maintaining such a high quality service. I have been a satisfied customer for too many years to count. While outside events ( an order seized by Customs) your company has kept every promise & made sure things were done to ensure delivery of products. I just want you to know that I can't think of any other company that is as excellent as Inhouse. The products offered are of top-notch quality. The customer service is incredibly effective & gracious in all communications. The updates on the order are wonderful, I know exactly how my order is moving thru the stages: order received/ order arranged for delivery/ order ready for mailing, tracking # given. It just hits all the check ✔️ marks. You folks blow other companies out of the water, just by doing things "right" & keeping communication lines open at every step.!! I appreciate you, & the other team members more than u will ever know. God Bless. "
Sandy Baker Michigian, USA • May 2026
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"I want to say a big thank you to everyone at Inhouse Pharmacy. Over the last 4 years, you have been such a valuable part of my life. You have listened to me, helped me and shown such kindness. It is not an exaggeration to say that without the supply of medication from yourselves, I would not be alive today. People like myself in the UK are literally left to our own devices as the medical industry denies us life critical care. Please keep up the good work, and help as many people as you can. Thank you for all your help. "
Alan UK • October 2024
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Cheryl Owens TX,USA • August 2025
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"Since 2003, Inhouse Pharmacy has continued to exceed my expectations of quality customer service. To date, I've experienced only one issue related to goods in transit, which was quickly remedied by Inhouse Pharmacy's customer service team. Whenever I have requested assistance from their staff, they have always been courteous, friendly and professional. I cannot fault their service. 10/10 stars, please keep doing what you are doing!"
Mateja NSW, AU • May 2026
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Kimberly NM, USA • August 2025
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"Hi, I just must stop and say thank you for all you girls have done over, the years. Your service is excellent! Always courteous and professional!"
David Koss PA, USA • July 2025
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"I have ordered with Inhouse for many years. They've always been excellent. Even after emergencies when we needed things in the past, I've never been let down. They've always been lovely to me and I just feel like I'm getting things from friends. So, I love Inhouse! There hasn't been anything bad, so it would be a new one if there ever was. The goods have always been delivered as seen and priced as advertised, and replaced if necessary. So, it's a straight 5-star award."
Gina UK • June 2026
 

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